Protein Details: KCa4.2 (Calcium-activated potassium channel)

Protein ID

ICDB_Pro_1119

Protein Name

KCa4.2 (Calcium-activated potassium channel)

Gene Name

Kcnt2; Slick

Organism

Rattus norvegicus (Rat)

Length

1142 amino acids

AlphaFoldDB

AF-Q6UVM4-F1-model_v4.pdb

Function

Outward rectifying potassium channel. Produces rapidly activating outward rectifier K(+) currents. Activated by high intracellular sodium and chloride levels . Channel activity is inhibited by ATP and by inhalation anesthetics; such as isoflurane. Inhibited upon stimulation of G-protein coupled receptors; such as CHRM1 and GRM1 (By similarity)

Sequence

MVDLESEVPPLPPRYRFRDLLLGDQGWQNDDRVQVEFYMNENTFKERLKLFFIKNQRSSLRIRLFNFSLKLLSCLLYIIRVLLEKPSQGNDWSHIFWVNRSLPLWGLQVSVALISLFETILLGYLSYKGNIWEQILRVPFILEIINAVPFIISIFWPTLRNLFVPVFLNCWLAKHALENMINDLHRAIQRTQSAMFNQVLILISTLLCLIFTCICGIQHLERIGKKLNLFDSLYFCIVTFSTVGFGDVTPETWSSKLFVVAMICVALVVLPIQFEQLAYLWMERQKSGGNYSRHRAQTEKHVVLCVSSLKIDLLMDFLNEFYAHPRLQDYYVVILCPTEMDVQVRRVLQIPMWSQRVIYLQGSALKDQDLLRAKMDNAEACFILSSRCEVDRTSSDHQTILRAWAVKDFAPNCPLYVQILKPENKFHIKFADHVVCEEEFKYAMLALNCICPATSTLITLLVHTSRGQCVCLCCREGQQSPEQWQKTYGRCSGNEVYHIVLEESTFFAEYEGKSFTYASFHAHKKFGVCLVGVRREDNKNILLNPGPRYIMNASDICFYINITKEENSAFKNQDQQRKSNVSRSFYHGPSRLPVHSIIASMGTVAIDLQDTSCRAASGPTLALPSEGGKELRRPSIAPVLEVADTSSIQTCDLLSDQSEDETTPDEETSSNLEYAKGYPPYSPYIGSSPTFCHLLQEKVPFCCLRLDKSCQHNYYEDAKAYGFKNKLIIVAAETAGNGLYNFIVPLRAYYRPKKELNPIVLLLDNPPDMHFLDAICWFPMVYYMVGSIDNLDDLLRCGVTFAANMVVVDKESTMSAEEDYMADAKTIVNVQTLFRLFSSLSIITELTHPANMRFMQFRAKDCYSLALSKLEKKERERGSNLAFMFRLPFAAGRVFSISMLDTLLYQSFVKDYMISITRLLLGLDTIPGSGFLCSMKITEDDLWIRTYARLYQKLCSSTGDVPIGIYRTESQKLTTSESQISISVEEWEDTKDVKDPGHHRSIHRNSTSSDQSDHPLLRRKSMQWARRLSRKGPKHSGKTAEKITQQRLNLYRRSERQELAELVKNRMKHLGLSTVGYDEMNDHQSTLSYILINPSPDTRLELNDVVYLIRPDPLSYLPNSEPSRKNSICNAAVQDSREETQL

PDB Structures

Ligand Binding

1. DICL_CP

2. DICL_Pep

Binding Site

1032..1039

Disease

Location

Detected in brain; and at low levels in heart. Detected in brainstem; including auditory neurons such as the medial nucleus of the trapezoid body. Detected in the olfactory bulb; red nucleus; facial nucleus; pontine nucleus; oculomotor nucleus; substantia nigra; deep cerebellar nuclei; vestibular nucleus; and the thalamus. Detected in hippocampal CA1; CA2; and CA3 regions; the dentate gyrus; supraoptic nucleus; hypothalamus; dorsal root ganglion; and cortical layers II; III; and V. Detected in striatum cholinergic interneurons.

DOI ID

10.1523/jneurosci.23-37-11681.2003; 10.1002/cne.20462; 10.1523/jneurosci.3372-05.2006; 10.1523/jneurosci.0551-07.2007; 10.1016/j.celrep.2017.09.088

RefSeq

NP_942057.1

Feature